K-252a - CAS# 99533-80-9 60261 2015 Jan 12

2015 Jan 12

InChi: InChI=1S/C10H11F3N2O5

GPR39-C3 was dosed to Male C57BL/6 mice via oral gavage at 30 mg/kg

Felbamate (W-554) is an anti-epileptic drug used in the treatment of epilepsy

is a potent and selective allosteric inhibitor of oncogenic K-Ras(G12C)

K-252a - CAS# 99533-80-9 60261 2015 Jan 12K 252a, CAS No. 99533 80 9, also known as SF 2370, is an alkaloid isolated from Nocardiopisis bacteria. This staurosporine analog is a highly potent cell permeable inhibitor of CaM kinase and phosphorylase kinase (IC50 = 1. 8 and 1. 7 nmol L, respectively). At higher concentrations it is also an efficient inhibitor of serine threonine protein kinases (IC50 of 10 to 30 nmol L). Product information CAS Number: 99533 80 9 Molecular Weight: 467. 47