Devazepide Catalog No.:M21854-C ML216 displays low micromolar potency

ML216 displays low micromolar potency and selectivity over related helicases

Regaloside A

injected intraperitoneally

7aR)-4-hydroxy-4-(m-tolylethynyl)octahydro-1H-indole-1-carboxylate

Smiles: NC1=CC2=C(C=C1)C1(OC2=O)C2=CC=C(O)C=C2OC2=CC(O)=CC=C12

Devazepide Catalog No.:M21854-C ML216 displays low micromolar potencyDevazepide (L 364,718) is a potent, competitive, selective and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor, with IC50s of 81 pM, 45 pM and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respectively. Devazepide (L 364,718) is effective for gastrointestinal disorders. Product information CAS Number: 103420 77 5 Molecular Weight: 408. 45 Formula: C25H20N4O2 Chemical Name: N [(3S) 1 methyl 2