![Raloxifene 4'-glucuronide 11377 dimethyl(2-{5-[(pyrrolidine-1-sulfonyl)methyl]-1H-indol-3-yl}ethyl)amine](https://cdn.shopify.com/s/files/1/0389/1897/9723/products/M14633_1631099723.gif?v=1631099725)
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dimethyl(2-{5-[(pyrrolidine-1-sulfonyl)methyl]-1H-indol-3-yl}ethyl)amine
is a specific inhibitor of the Ca(2+)/calmodulin-dependent protein kinase kinase
7 inhibitor
thereby prolonging repolarization
InChiKey: HGWLTZOMQZIUBW-UHFFFAOYSA-N
Raloxifene 4'-glucuronide 11377 dimethyl(2-{5-[(pyrrolidine-1-sulfonyl)methyl]-1H-indol-3-yl}ethyl)amineRaloxifene 4' glucuronide is a primary metabolite of Raloxifene. Raloxifene 4' glucuronide formation is mediated mostly by UGT1A10 and UGT1A8. Raloxifene 4' glucuronide binds to estrogen receptor with an IC50 of 370 M. . Raloxifene is a selective estrogen receptor modulator. Raloxifene activates TGF3 promoter as a full agonist at nanomolar concentrations, and inhibits the estrogen response element containing vitellogenin promoter expression. Product
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